Search results for: 'Protein Tyrosine Kinase'

Cat. No.	Name	CAS No.	Description
KI1195	BMS777607	1196681-44-3	BMS777607 is a selective and orally efficacious inhibitor of the Met kinase superfamily....
KI4990	BMS-794833	1174046-72-0	....
KI3420	BMS-554417	468741-42-6	BMS-554417 is a inhibitor of IGF1R/IR and inhibits focal adhesion kinase (FAK) activity....
KI0425	BMS-536924	468740-43-4	BMS-536924 is a novel small-molecule inhibitor which prevents activity of the insulin-like growth factor receptor kinase....
KI0068	BIBW2992	439081-18-2	BIBW2992 is an irreversible inhibitor of ErbB family with IC50s of 0.5, 14 and 1 nM for epidermal growth factor receptor (EGFR) (ErbB1/HER1), HER2 and HER4 kinases....
KI0195	BIBF1120	656247-17-5	BIBF1120 is a potent vascular endothelial growth factor receptor (VEGFR), platelet-derived growth factor receptors (PDGFR) and fibroblast growth factor receptors (FGFR) kinase inhibitor....
KI1151	BGJ398	872511-34-7	BGJ398 is a potent and selective inhibitor of the FGFR family of tyrosine kinase receptors FGFR1, FGFR2, FGFR3, and FGFR4 with IC50s of 0.9, 1.4, 1 and 60 nM, respectively....
KI1303	AZD8931	848942-61-0	AZD8931 is a reversible, ATP competitive inhibitor of epidermal growth factor receptor (EGFR; erbB1), erbB2 (human epidermal growth factor receptor 2), and erbB3 receptor with IC50 of 4, 3 and 4 nM, respectively....
KI0595	AZD4547	1035270-39-3	AZD4547 is a potent selective FGFR inhibitor....
KI3677	AZD3463	1356962-20-3	....
KI3884	AZD2858	486424-20-8	....
KI0269	AZD1480	935666-88-9	AZD1480 is a potent ATP competitive inhibitor of JAK2 kinase, with an inhibition constant (K_{i) of 0.26 nM....}
KI0443	Axitinib	319460-85-0	Axitinib is a potent and selective inhibitor of VEGF receptor tyrosine kinase (RTK) 1, 2, and 3....
KI2617	AVL-292	1202757-89-8	AVL-292 is a selective and covalent inhibitor of Bruton's tyrosine kinase (Btk)....
KI3415	AV-412	451493-31-5	AV-412 is a potent dual inhibitor of epidermal growth factor receptor (EGFR) and ErbB2 tyrosine kinases, including the mutant EGFRL858R,T790M....
KI2814	ARQ-197	905854-02-6	ARQ-197 is the first non-ATP-competitive and selective c-Met receptor inhibitor....
KI4027	Apixaban	503612-47-3	....
KI3645	Apatinib	811803-05-1	Apatinib, also known as YN968D1, is a tyrosine kinase inhibitor that selectively inhibits the vascular endothelial growth factor receptor-2 (VEGFR2, also known as KDR) with IC50 of 1nM ^[1]....
KI4885	AP26113	1197958-12-5	....
KI1465	AMG458	913376-83-7	AMG458 is a novel selective c-Met inhibitor....