Cat. No. |
Name |
CAS No. |
Description |
KI3077 |
ZSTK474 |
475110-96-4 |
ZSTK474 is an ATP-competitive pan-class I PI3K inhibitor....
|
KI0339 |
XL765(SAR-245409) |
1349796-36-6 |
XL765 is a small molecule dual-targeted PI3K/mTOR inhibitor, which inhibits PI3Kα, PI3Kβ, PI3Kδ and PI3Kγwith IC50 values of 39, 113, 43 and 9 nM, respectively....
|
KI3070 |
XL147(SAR245408) |
956958-53-5 |
XL147 (SAR245408) is a PI3K inhibitor....
|
KI3098 |
XL-765 (SAR-245409) |
1123889-87-1 |
XL765 is a potent and selective inhibitor of Class I PI3K isoforms and mTOR....
|
KI0545 |
WYE-687 |
1062161-90-3 |
WYE-687 is a potent and ATP-competitive inhibitor of mTOR....
|
KI0542 |
WYE-354 |
1062169-56-5 |
WYE-354 is a potent and ATP-competitive inhibitor of mTOR....
|
KI1444 |
WYE-125132 |
1144068-46-1 |
WYE-125132 is a highly potent, ATP-competitive, and specific mTOR kinase inhibitor....
|
KI0538 |
WAY-600 |
1062159-35-6 |
WAY-600 is a potent and ATP-competitive inhibitor of mTOR....
|
KI0865 |
VS-5584 |
1246560-33-7 |
VS-5584 is a selective dual PI3K/mTOR inhibitor that potently inhibits mTOR kinase PI3K isoforms....
|
KI4136 |
TWS119 |
601514-19-6 |
....
|
KI0128 |
Triciribine |
35943-35-2 |
Triciribine is a potent Akt inhibitor with IC50 of 130 nM....
|
KI3941 |
TPCA1 |
507475-17-4 |
....
|
KI0617 |
Torin2 |
1223001-51-1 |
Torin 2 is a potent, selective and orally available mTOR inhibitor....
|
KI0010 |
TGX-221 |
663619-89-4 |
TGX-221 is a potent and selective phosphoinositide 3-kinase (PI3K) p110β inhibitor with an IC50 of 8.5 nM....
|
KI0244 |
Temsirolimus |
162635-04-3 |
Temsirolimus is a specific inhibitor of mTOR used in the treatment of renal cell carcinoma....
|
KI0494 |
SB 415286 |
264218-23-7 |
SB 415286 is a potent and selective cell permeable glycogen synthase kinase 3 (GSK3) inhibitor....
|
KI3330 |
SB 216763 |
280744-09-4 |
SB 216763 is a potent, selective, and ATP-competitive inhibitor of glycogen synthase kinase-3 (GSK-3)....
|
KI0298 |
Rapamycin |
53123-88-9 |
Rapamycin forms a complex with FK506-binding protein 12 that binds and inhibits mammalian target of TOR kinase activity, leading to dephosphorylation of downstream targets of mTOR, S6K1, and 4E-BP1....
|
KI2091 |
PX-866 |
502632-66-8 |
PX-866, a derivative of wortmannin, is a potent PI3 Kinase inhibitor....
|
KI0549 |
PP242 |
1092351-67-1 |
PP242 is a mammalian target of rapamycin (mTOR) inhibitor....
|