Cat. No. |
Name |
CAS No. |
Description |
KI0199 |
AC220 |
950769-58-1 |
AC220 is a unique, potent and selective inhibitor of fms-like tyrosine kinase (FLT3) with IC50 values of 1.1 and 4.2 nM for internal tandem duplications mutation FLT3 (FLT3-ITD) and wild type FLT3 (FLT3-WT) autophosphorylation, respectively....
|
KI1299 |
AEE788 |
497839-62-0 |
AEE788 is a novel multitargeted inhibitor of EGFR, ErbB2, KDR, and Flt-1 with IC50 values of 2, 6, 77 and 59 nM, respectively....
|
KI6066 |
AG 18 |
118409-57-7 |
....
|
KI3495 |
AG-1024 |
65678-07-1 |
AG1024 is an IGF-1R inhibitor....
|
KI0514 |
AG-1478 |
153436-53-4 |
AG-1478 is an inhibitor of the EGFR tyrosine kinase....
|
KI0512 |
AG-490 |
133550-30-8 |
AG-490 is a specific janus kinase 2 (JAK2) inhibitor....
|
KI0465 |
AG879 |
148741-30-4 |
AG 879 is widely used specific Tyr kinase inhibitor for ErbB2 and FLK-1 (a VEGF receptor)....
|
KI6085 |
Altiratinib |
1345847-93-9 |
....
|
KI2800 |
AMG-208 |
1002304-34-8 |
AMG 208 is a potent and selective inhibitor of kinase c-Met....
|
KI1465 |
AMG458 |
913376-83-7 |
AMG458 is a novel selective c-Met inhibitor....
|
KI4885 |
AP26113 |
1197958-12-5 |
....
|
KI3645 |
Apatinib |
811803-05-1 |
Apatinib, also known as YN968D1, is a tyrosine kinase inhibitor that selectively inhibits the vascular endothelial growth factor receptor-2 (VEGFR2, also known as KDR) with IC50 of 1nM [1]....
|
KI4027 |
Apixaban |
503612-47-3 |
....
|
KI2814 |
ARQ-197 |
905854-02-6 |
ARQ-197 is the first non-ATP-competitive and selective c-Met receptor inhibitor....
|
KI3415 |
AV-412 |
451493-31-5 |
AV-412 is a potent dual inhibitor of epidermal growth factor receptor (EGFR) and ErbB2 tyrosine kinases, including the mutant EGFRL858R,T790M....
|
KI2617 |
AVL-292 |
1202757-89-8 |
AVL-292 is a selective and covalent inhibitor of Bruton's tyrosine kinase (Btk)....
|
KI0443 |
Axitinib |
319460-85-0 |
Axitinib is a potent and selective inhibitor of VEGF receptor tyrosine kinase (RTK) 1, 2, and 3....
|
KI0269 |
AZD1480 |
935666-88-9 |
AZD1480 is a potent ATP competitive inhibitor of JAK2 kinase, with an inhibition constant (Ki) of 0.26 nM....
|
KI3884 |
AZD2858 |
486424-20-8 |
....
|
KI3677 |
AZD3463 |
1356962-20-3 |
....
|