| Cat. No. |
Name |
CAS No. |
Description |
|
KI0629 |
Gsk1904529A |
1089283-49-7 |
GSK1904529A is a small-molecule inhibitor of the insulin-like growth factor-I receptor tyrosine kinase....
|
|
KI3962 |
GSK256066 |
801312-28-7 |
....
|
|
KI3455 |
GW 441756 |
504433-23-2 |
GW441756 is a potent and selective inhibitor of the NGF receptor tyrosine kinase A (TrkA)....
|
|
KI5003 |
GW2580 |
870483-87-7 |
....
|
|
KI0301 |
Imatinib |
152459-95-5 |
Imatinib is a 2-phenylaminopyrimidine derivative that functions as a multi-target inhibitor of tyrosine kinase enzymes with IC50 values of 0.6, 0.1 and 0.1 μM for v-Abl, c-kit and PDGFR, respectively....
|
|
KI4317 |
Imatinib Mesylate |
220127-57-1 |
....
|
|
KI0207 |
INCB018424 |
941678-49-5 |
INCB018424 is a potent and selective inhibitor of JAK1 (Janus kinase) and JAK2 with IC50 of 3.3 and 2.8 nM, respectively....
|
|
KI0632 |
INCB28060 |
1029712-80-8 |
INCB28060 is a novel inhibitor of c-MET kinase....
|
|
KI0420 |
JNJ-38877605 |
943540-75-8 |
JNJ-38877605 is a small-molecule, ATP-competitive inhibitor of the catalytic activity of c-Met....
|
|
KI3335 |
KRN 633 |
286370-15-8 |
KRN 633 is a novel quinazoline urea derivative and a potent ATP-competitive inhibitor of VEGFR-1, -2 and -3 with IC50s of 170, 160, and 125 nM, respectively....
|
|
KI0431 |
Lapatinib |
231277-92-2 |
Lapatinib is a selective inhibitor of both epidermal growth factor receptor (EGFR) and HER-2 tyrosine kinases with IC50 of 10.2 and 9.8 nM, respectively....
|
|
KI4179 |
LDK378 |
1032900-25-6 |
....
|
|
KI1019 |
Lestaurtinib |
111358-88-4 |
Lestaurtinib is a potent and orally available fms-like kinase (FLT3) inhibitor....
|
|
KI0047 |
Linifanib |
796967-16-3 |
Linifanib is a receptor tyrosine kinase (RTK) inhibitor....
|
|
KI0380 |
LY2784544 |
1229236-86-5 |
LY2784544 has been identified as being highly selective for JAK 2-V617F and has advanced into human clinical trials for the treatment of several myeloproliferative disorders....
|
|
KI1453 |
LY2801653 |
1206799-15-6 |
LY2801653 is a type-II ATP competitive, slow-off inhibitor of MET tyrosine kinase....
|
|
KI4071 |
LY2811376 |
1194044-20-6 |
....
|
|
KI1359 |
Masitinib |
790299-79-5 |
Masitinib is a potent and selective inhibitor of KIT....
|
|
KI4704 |
MK-2461 |
917879-39-1 |
....
|
|
KI2821 |
MK-8033 |
1196681-38-5 |
MK-8033 is a dual c-Met/Ron inhibitor....
|
