| Cat. No. |
Name |
CAS No. |
Description |
|
KI0637 |
AS703026 |
1236699-92-5 |
AS703026 is a novel, selective, orally bioavailable mitogen-activated protein kinase (MEK) 1/2 inhibitor, in human multiple myeloma (MM)....
|
|
KI1330 |
AZD6244 |
606143-52-6 |
AZD6244 is a potent, selective, and ATP-uncompetitive inhibitor of MEK1/2 kinases....
|
|
KI6051 |
B-Raf IN 1 |
950736-05-7 |
....
|
|
KI0473 |
BIX 02188 |
1094614-84-2 |
BIX02188 is a selective and potent MEK5 inhibitor....
|
|
KI0477 |
BIX 02189 |
1094614-85-3 |
BIX02189 is a selective and potent MEK5 inhibitor....
|
|
KI0556 |
CCT239065 |
1163719-51-4 |
CCT239065 is a BRAFV600E inhibitor....
|
|
KI2349 |
CEP-32496 |
1188910-76-0 |
CEP-32496 is a potent BRAF inhibitor....
|
|
KI0387 |
CI-1040 |
212631-79-3 |
CI-1040 is a small-molecule with highly selective adenosine triphosphate (ATP) non-competitive inhibition activity against MEK1/2....
|
|
KI2068 |
CPI-613 |
95809-78-2 |
CPI-613 is a non-redox active lipoate derivative that selectively inhibits mitochondrial enzymes pyruvate dehydrogenase (PDH) and α-ketoglutarate dehydrogenase....
|
|
KI4996 |
Dabrafenib |
1195765-45-7 |
....
|
|
KI2791 |
Dabrafenib Mesylate |
1195768-06-9 |
Dabrafenib mesylate is a mutant-BRAF kinase inhibitor....
|
|
KI6137 |
DB07268 |
929007-72-7 |
....
|
|
KI1395 |
Doramapimod |
285983-48-4 |
Doramapimod is a picomolar inhibitor of human p38 MAP kinase with Kγ of 0.1 nM....
|
|
KI0311 |
GDC-0879 |
905281-76-7 |
GDC-0879 is a highly selective and orally bioavailable RAF small-molecule inhibitor....
|
|
KI1165 |
GSK1120212 |
871700-17-3 |
GSK1120212 is a selective and highly potent MEK1 and MEK2 inhibitor with IC50 values of 1.8 and 0.92 nM, respectively....
|
|
KI5005 |
JNK-IN-8 |
1410880-22-6 |
....
|
|
KI0260 |
LY2228820 |
862507-23-1 |
LY2228820 is a novel p38 mitogen-activated protein kinase (p38MAPK) inhibitor....
|
|
KI0289 |
Nilotinib |
641571-10-0 |
Nilotinib inhibits the kinases BCR-ABL, KIT, LCK, EPHA3, EPHA8, DDR1, DDR2, PDGFRB, MAPK11 and ZAK....
|
|
KI0357 |
PD0325901 |
391210-10-9 |
PD0325901 is selective and non ATP-competitive mitogenic extracellular kinase 1/2 (MEK1/2) inhibitor with an IC50 of 0.33 nM....
|
|
KI3370 |
PD318088 |
391210-00-7 |
PD318088 is a non-ATP competitive MEK inhibitor....
|
