Cat. No. |
Name |
CAS No. |
Description |
KI1124 |
TG101348 |
936091-26-8 |
TG101348 is a selective small-molecule inhibitor of JAK2....
|
KI1173 |
TG101209 |
936091-14-4 |
TG101209 potently inhibits JAK2, FLT3 and RET kinases with IC50 values of 6, 25 and 17 nM, respectively....
|
KI1113 |
Telatinib |
332012-40-5 |
Telatinib is an orally available, small-molecule multitargeted vascular endothelial growth factor receptors 2 and 3 (VEGFR-2/-3) and platelet-derived growth factor receptor β tyrosine kinases inhibitor....
|
KI2104 |
TCS 401 |
243967-42-2 |
TCS 401 is a selective inhibitor of protein-tyrosine phosphatase 1B (PTP1B) with a Ki value of 290 nM....
|
KI1270 |
TAE684 |
761439-42-3 |
TAE684 is a potent ALK inhibitor with an IC50 of 3 nM....
|
KI0234 |
Sunitinib |
557795-19-4 |
Sunitinib is a multitargeted kinase inhibitor that inhibits vascular endothelial growth factor receptor (VEGFR) -1, 2 and 3, platelet-derived growth factor receptors (PDGFR)-α and β, Flt3 (Fms-like tyrosyl kinase-3), Ret, and Kit....
|
KI4773 |
SU5416 |
204005-46-9 |
....
|
KI2718 |
SU14813 |
627908-92-3 |
SU14813 is a novel multiple receptor tyrosine kinase inhibitor....
|
KI0107 |
Su11274 |
658084-23-2 |
Su11274 is a ATP-competitive c-Met specific inhibitor....
|
KI3305 |
SU 5402 |
215543-92-3 |
SU5402 is a potent and selective inhibitor of vascular endothelial growth factor receptor (VEGFR) and fibroblast growth factor receptor (FGFR)....
|
KI4000 |
SKLB1002 |
1225451-84-2 |
....
|
KI1266 |
SGX-523 |
1022150-57-7 |
SGX-523 is a potent and selective Met inhibitor with an IC50 of 4 nM....
|
KI3937 |
SCH727965 |
779353-01-4 |
....
|
KI3360 |
SB 525334 |
356559-20-1 |
SB525334 is a potent and selective inhibitor of the transforming growth factor-β1 (TGF-β1) receptor (ALK5)....
|
KI0136 |
SB 431542 |
301836-41-9 |
SB-431542 is a novel, small molecule ATP-mimetic inhibitor of the kinase activity associated with members of the activin receptor-like kinase (ALK) family-specifically ALK5 (TGF- β type I receptor, TGF- β RI), ALK4 (activin type I receptor), and ALK7 (nodal type I receptor)....
|
KI0072 |
Saracatinib |
379231-04-6 |
Saracatinib is a novel Src family kinase/Abl dual-kinase inhibitor for c-Src and v-Abl with IC50 values of 2.7 and 30 nM, respectively....
|
KI2505 |
RN486 |
1242156-23-5 |
RN486 is a potent, selectively and proprietary Bruton's tyrosine kinase (Btk) inhibitor....
|
KI1326 |
Regorafenib |
755037-03-7 |
Regorafenib is an oral multi-kinase inhibitor....
|
KI0013 |
RAF265 |
927880-90-8 |
RAF265 is a selective and potent inhibitor of RAF and VEGFR2....
|
KI0098 |
R935788 |
1025687-58-4 |
Fostamatinib is the prodrug of R406, a specific ATP-competitive spleen tyrosine kinase (SYK) inhibitor with an IC50 of 41 nM....
|