| Cat. No. |
Name |
CAS No. |
Description |
|
KI0211 |
R406 |
841290-81-1 |
R406 is an ATP-competitive inhibitor of spleen tyrosine kinase (Syk) kinase with an IC50 of 41 nM....
|
|
KI2368 |
PRT062607 (P505-15, BIIB057) HCl |
1370261-97-4 |
PRT062607 is a novel, highly selective, and orally bioavailable small molecule spleen tyrosine kinase (SYK) inhibitor with an IC50 of 1 nM....
|
|
KI4891 |
PQ 401 |
196868-63-0 |
....
|
|
KI3953 |
PP121 |
1092788-83-4 |
....
|
|
KI3590 |
PKC412(midostaurin) |
120685-11-2 |
PKC412 is a selective protein kinase C (PKC) inhibitor....
|
|
KI1169 |
PHA-665752 |
477575-56-7 |
PHA-665752 is a potent, ATP-competitive inhibitor of c-Met kinase with an IC50 of 9 nM and Ki value of 4 nM....
|
|
KI1063 |
PF299804 |
1110813-31-4 |
PF299804 is an irreversible Pan-ERBB inhibitor....
|
|
KI2575 |
PF06465469 |
1407966-77-1 |
PF-06465469 is a potent inhibitor of interleukin-2 inducible T cell kinase (ITK)....
|
|
KI0017 |
PF-04217903 |
956905-27-4 |
PF-04217903 is a novel ATP-competitive small-molecule inhibitor of c-Met kinase....
|
|
KI2372 |
PD173955 |
260415-63-2 |
PD173955 is a Src family-specific tyrosine kinase inhibitor....
|
|
KI0248 |
PD173074 |
219580-11-7 |
PD173074 is an ATP pocket inhibitor that inhibits the tyrosine kinase activities of the FGF and VEGF receptors....
|
|
KI4709 |
PD168393 |
194423-15-9 |
....
|
|
KI1436 |
PD153035 HCl |
183322-45-4 |
PD153035 is a specific and potent inhibitor of the epidermal growth factor (EGF) receptor tyrosine kinase....
|
|
KI2697 |
PCI-32765(ibrutinib) |
936563-96-1 |
PCI-32765 is a selective and covalent inhibitor of Bruton's tyrosine kinase (Btk)....
|
|
KI0307 |
Pazopanib |
444731-52-6 |
Pazopanib is a novel orally available, small-molecule tyrosine kinase inhibitor of VEGF receptor (VEGFR) -1, -2, -3, PDGFR-α, PDGFR-β, and c-Kit with IC50 values of 10, 30, 47, 71, 84 and 74 nM, respectively....
|
|
KI1293 |
Pacritinib |
937272-79-2 |
Pacritinib is a novel oral JAK2 inhibitor....
|
|
KI4399 |
OSI930 |
728033-96-3 |
....
|
|
KI0172 |
Osi-906 |
867160-71-2 |
Osi-906 is a selective and orally efficacious dual inhibitor of the IGF-1 (insulin-like growth factor 1) receptor and insulin receptor (IR)....
|
|
KI0123 |
NVP-BVU972 |
1185763-69-2 |
NVP-BVU972 is a selective and potent MET kinase inhibitor with IC50 of 14 nM....
|
|
KI3702 |
NVP-BSK805 dihydrochloride |
1092499-93-8 |
NVP-BSK805 can potently suppress JAK2 with IC50 of 0.5 nM, and displays more than 20-fold selectivity towards JAK1, JAK3, and TYK2....
|
