| Cat. No. |
Name |
CAS No. |
Description |
|
KI0017 |
PF-04217903 |
956905-27-4 |
PF-04217903 is a novel ATP-competitive small-molecule inhibitor of c-Met kinase....
|
|
KI2575 |
PF06465469 |
1407966-77-1 |
PF-06465469 is a potent inhibitor of interleukin-2 inducible T cell kinase (ITK)....
|
|
KI1063 |
PF299804 |
1110813-31-4 |
PF299804 is an irreversible Pan-ERBB inhibitor....
|
|
KI1169 |
PHA-665752 |
477575-56-7 |
PHA-665752 is a potent, ATP-competitive inhibitor of c-Met kinase with an IC50 of 9 nM and Ki value of 4 nM....
|
|
KI3590 |
PKC412(midostaurin) |
120685-11-2 |
PKC412 is a selective protein kinase C (PKC) inhibitor....
|
|
KI3953 |
PP121 |
1092788-83-4 |
....
|
|
KI4891 |
PQ 401 |
196868-63-0 |
....
|
|
KI2368 |
PRT062607 (P505-15, BIIB057) HCl |
1370261-97-4 |
PRT062607 is a novel, highly selective, and orally bioavailable small molecule spleen tyrosine kinase (SYK) inhibitor with an IC50 of 1 nM....
|
|
KI0211 |
R406 |
841290-81-1 |
R406 is an ATP-competitive inhibitor of spleen tyrosine kinase (Syk) kinase with an IC50 of 41 nM....
|
|
KI0098 |
R935788 |
1025687-58-4 |
Fostamatinib is the prodrug of R406, a specific ATP-competitive spleen tyrosine kinase (SYK) inhibitor with an IC50 of 41 nM....
|
|
KI0013 |
RAF265 |
927880-90-8 |
RAF265 is a selective and potent inhibitor of RAF and VEGFR2....
|
|
KI1326 |
Regorafenib |
755037-03-7 |
Regorafenib is an oral multi-kinase inhibitor....
|
|
KI2505 |
RN486 |
1242156-23-5 |
RN486 is a potent, selectively and proprietary Bruton's tyrosine kinase (Btk) inhibitor....
|
|
KI0072 |
Saracatinib |
379231-04-6 |
Saracatinib is a novel Src family kinase/Abl dual-kinase inhibitor for c-Src and v-Abl with IC50 values of 2.7 and 30 nM, respectively....
|
|
KI0136 |
SB 431542 |
301836-41-9 |
SB-431542 is a novel, small molecule ATP-mimetic inhibitor of the kinase activity associated with members of the activin receptor-like kinase (ALK) family-specifically ALK5 (TGF- β type I receptor, TGF- β RI), ALK4 (activin type I receptor), and ALK7 (nodal type I receptor)....
|
|
KI3360 |
SB 525334 |
356559-20-1 |
SB525334 is a potent and selective inhibitor of the transforming growth factor-β1 (TGF-β1) receptor (ALK5)....
|
|
KI3937 |
SCH727965 |
779353-01-4 |
....
|
|
KI1266 |
SGX-523 |
1022150-57-7 |
SGX-523 is a potent and selective Met inhibitor with an IC50 of 4 nM....
|
|
KI4000 |
SKLB1002 |
1225451-84-2 |
....
|
|
KI3305 |
SU 5402 |
215543-92-3 |
SU5402 is a potent and selective inhibitor of vascular endothelial growth factor receptor (VEGFR) and fibroblast growth factor receptor (FGFR)....
|
