| Cat. No. |
Name |
CAS No. |
Description |
|
KI4147 |
NVP-BHG712 |
940310-85-0 |
....
|
|
KI1334 |
NVP-AEW541 |
475489-16-8 |
NVP-AEW541 is a novel, potent, and selective inhibitor of the IGF-IR kinase....
|
|
KI3430 |
NVP-ADW742 |
475488-23-4 |
NVP-ADW742 is a small molecule ATP-competitive inhibitor of the IGF-I receptor (IGF-IR) with an IC50 of 0.17 µM....
|
|
KI2103 |
NSC 87877 |
56990-57-9 |
NSC 87877 is a potent inhibitor of shp2 and shp1 protein tyrosine phosphatases (PTP)....
|
|
KI0289 |
Nilotinib |
641571-10-0 |
Nilotinib inhibits the kinases BCR-ABL, KIT, LCK, EPHA3, EPHA8, DDR1, DDR2, PDGFRB, MAPK11 and ZAK....
|
|
KI0084 |
Neratinib |
698387-09-6 |
Neratinib is a dual inhibitor of the human epidermal growth factor receptor 2 (HER2) and epidermal growth factor receptor (EGFR) kinases....
|
|
KI4363 |
Nelarabine |
121032-29-9 |
....
|
|
KI0275 |
MP-470 |
850879-09-03 |
MP-470 is a novel orally bioavailable mutitargeting tyrosine kinase inhibitor with activity against mutant c-KIT, PDGFRa and FLT3....
|
|
KI4665 |
Motesanib |
453562-69-1 |
....
|
|
KI2821 |
MK-8033 |
1196681-38-5 |
MK-8033 is a dual c-Met/Ron inhibitor....
|
|
KI4704 |
MK-2461 |
917879-39-1 |
....
|
|
KI1359 |
Masitinib |
790299-79-5 |
Masitinib is a potent and selective inhibitor of KIT....
|
|
KI4071 |
LY2811376 |
1194044-20-6 |
....
|
|
KI1453 |
LY2801653 |
1206799-15-6 |
LY2801653 is a type-II ATP competitive, slow-off inhibitor of MET tyrosine kinase....
|
|
KI0380 |
LY2784544 |
1229236-86-5 |
LY2784544 has been identified as being highly selective for JAK 2-V617F and has advanced into human clinical trials for the treatment of several myeloproliferative disorders....
|
|
KI0047 |
Linifanib |
796967-16-3 |
Linifanib is a receptor tyrosine kinase (RTK) inhibitor....
|
|
KI1019 |
Lestaurtinib |
111358-88-4 |
Lestaurtinib is a potent and orally available fms-like kinase (FLT3) inhibitor....
|
|
KI4179 |
LDK378 |
1032900-25-6 |
....
|
|
KI0431 |
Lapatinib |
231277-92-2 |
Lapatinib is a selective inhibitor of both epidermal growth factor receptor (EGFR) and HER-2 tyrosine kinases with IC50 of 10.2 and 9.8 nM, respectively....
|
|
KI3335 |
KRN 633 |
286370-15-8 |
KRN 633 is a novel quinazoline urea derivative and a potent ATP-competitive inhibitor of VEGFR-1, -2 and -3 with IC50s of 170, 160, and 125 nM, respectively....
|
