| Cat. No. |
Name |
CAS No. |
Description |
|
KI0420 |
JNJ-38877605 |
943540-75-8 |
JNJ-38877605 is a small-molecule, ATP-competitive inhibitor of the catalytic activity of c-Met....
|
|
KI0632 |
INCB28060 |
1029712-80-8 |
INCB28060 is a novel inhibitor of c-MET kinase....
|
|
KI0207 |
INCB018424 |
941678-49-5 |
INCB018424 is a potent and selective inhibitor of JAK1 (Janus kinase) and JAK2 with IC50 of 3.3 and 2.8 nM, respectively....
|
|
KI4317 |
Imatinib Mesylate |
220127-57-1 |
....
|
|
KI0301 |
Imatinib |
152459-95-5 |
Imatinib is a 2-phenylaminopyrimidine derivative that functions as a multi-target inhibitor of tyrosine kinase enzymes with IC50 values of 0.6, 0.1 and 0.1 μM for v-Abl, c-kit and PDGFR, respectively....
|
|
KI5003 |
GW2580 |
870483-87-7 |
....
|
|
KI3455 |
GW 441756 |
504433-23-2 |
GW441756 is a potent and selective inhibitor of the NGF receptor tyrosine kinase A (TrkA)....
|
|
KI3962 |
GSK256066 |
801312-28-7 |
....
|
|
KI0629 |
Gsk1904529A |
1089283-49-7 |
GSK1904529A is a small-molecule inhibitor of the insulin-like growth factor-I receptor tyrosine kinase....
|
|
KI0552 |
GSK1838705A |
1116235-97-2 |
GSK1838705A is a small-molecule IGF-IR and the insulin receptor inhibitor....
|
|
KI3963 |
GSK1349572 |
1051375-16-6 |
....
|
|
KI0309 |
Gefitinib |
184475-35-2 |
Gefitinib, a synthetic anilinoquinazoline, directly and specificly inhibits tyrosine kinase (TK) phosphorylation on the epidermal growth factor receptor (EGFR) by competing for the ATP-binding site, which leads to suppression of the EGFR pathway (HER-kinase axis)....
|
|
KI6095 |
FLT3-IN-1 |
1370256-78-2 |
....
|
|
KI2647 |
FLLL32 |
1226895-15-3 |
FLLL32 is a novel and small molecule inhibitor of the STAT3 pathway....
|
|
KI4041 |
Fasudil hydrochloride |
105628-07-7 |
....
|
|
KI0303 |
Erlotinib Hydrochloride |
183319-69-9 |
Erlotinib is a selective, orally available small-molecule inhibitor of the HER1/EGFR tyrosine kinase domain, used to treat non-small cell lung cancer, pancreatic cancer and several other types of cancer....
|
|
KI3882 |
EPZ004777 |
1338466-77-5 |
....
|
|
KI2807 |
EMD-1214063 |
1100598-32-0 |
EMD-1214063 is a potent and selective inhibitor of c-Met....
|
|
KI3395 |
E7080 (Lenvatinib) |
417716-92-8 |
E7080 is an orally active inhibitor of multiple receptor tyrosine kinases, mostly for VEGFR2 (KDR)/VEGFR3 (Flt-4)....
|
|
KI2658 |
E-7050 |
928037-13-2 |
E-7050 is novel small molecule inhibitor of the c-Met and VEGFR-2 tyrosine kinases....
|
