Cat. No. |
Name |
CAS No. |
Description |
KI4665 |
Motesanib |
453562-69-1 |
....
|
KI0275 |
MP-470 |
850879-09-03 |
MP-470 is a novel orally bioavailable mutitargeting tyrosine kinase inhibitor with activity against mutant c-KIT, PDGFRa and FLT3....
|
KI4363 |
Nelarabine |
121032-29-9 |
....
|
KI0084 |
Neratinib |
698387-09-6 |
Neratinib is a dual inhibitor of the human epidermal growth factor receptor 2 (HER2) and epidermal growth factor receptor (EGFR) kinases....
|
KI0289 |
Nilotinib |
641571-10-0 |
Nilotinib inhibits the kinases BCR-ABL, KIT, LCK, EPHA3, EPHA8, DDR1, DDR2, PDGFRB, MAPK11 and ZAK....
|
KI2103 |
NSC 87877 |
56990-57-9 |
NSC 87877 is a potent inhibitor of shp2 and shp1 protein tyrosine phosphatases (PTP)....
|
KI3430 |
NVP-ADW742 |
475488-23-4 |
NVP-ADW742 is a small molecule ATP-competitive inhibitor of the IGF-I receptor (IGF-IR) with an IC50 of 0.17 µM....
|
KI1334 |
NVP-AEW541 |
475489-16-8 |
NVP-AEW541 is a novel, potent, and selective inhibitor of the IGF-IR kinase....
|
KI4147 |
NVP-BHG712 |
940310-85-0 |
....
|
KI3702 |
NVP-BSK805 dihydrochloride |
1092499-93-8 |
NVP-BSK805 can potently suppress JAK2 with IC50 of 0.5 nM, and displays more than 20-fold selectivity towards JAK1, JAK3, and TYK2....
|
KI0123 |
NVP-BVU972 |
1185763-69-2 |
NVP-BVU972 is a selective and potent MET kinase inhibitor with IC50 of 14 nM....
|
KI0172 |
Osi-906 |
867160-71-2 |
Osi-906 is a selective and orally efficacious dual inhibitor of the IGF-1 (insulin-like growth factor 1) receptor and insulin receptor (IR)....
|
KI4399 |
OSI930 |
728033-96-3 |
....
|
KI1293 |
Pacritinib |
937272-79-2 |
Pacritinib is a novel oral JAK2 inhibitor....
|
KI0307 |
Pazopanib |
444731-52-6 |
Pazopanib is a novel orally available, small-molecule tyrosine kinase inhibitor of VEGF receptor (VEGFR) -1, -2, -3, PDGFR-α, PDGFR-β, and c-Kit with IC50 values of 10, 30, 47, 71, 84 and 74 nM, respectively....
|
KI2697 |
PCI-32765(ibrutinib) |
936563-96-1 |
PCI-32765 is a selective and covalent inhibitor of Bruton's tyrosine kinase (Btk)....
|
KI1436 |
PD153035 HCl |
183322-45-4 |
PD153035 is a specific and potent inhibitor of the epidermal growth factor (EGF) receptor tyrosine kinase....
|
KI4709 |
PD168393 |
194423-15-9 |
....
|
KI0248 |
PD173074 |
219580-11-7 |
PD173074 is an ATP pocket inhibitor that inhibits the tyrosine kinase activities of the FGF and VEGF receptors....
|
KI2372 |
PD173955 |
260415-63-2 |
PD173955 is a Src family-specific tyrosine kinase inhibitor....
|